Journal article icon

Journal article

Pentamethylphenyl (Ph*) ketones: Unique building blocks for organic synthesis

Abstract:
Pentamethylphenyl (Ph*) ketones are rapidly emerging as versatile and useful building blocks for organic synthesis. The ortho-methyl substituents force the aromatic ring to twist out of planarity with the carbonyl, and consequently these molecules display a unique pattern of reactivity which is completely distinct to that of traditional aromatic ketones. The primary aim of this Digest is to highlight examples where new chemical reactivity is unlocked through the use of Ph* ketones, and a wide range of examples are presented including hydrogen borrowing catalysis, aldol addition and organocatalysis. Finally, methods to cleave the Ph* group to a range of other functionality are surveyed.
Publication status:
Published
Peer review status:
Peer reviewed

Actions


Access Document


Publisher copy:
10.1016/j.tetlet.2021.153151

Authors


More by this author
Institution:
University of Oxford
Division:
MPLS
Department:
Chemistry
Sub department:
Organic Chemistry
Role:
Author


Publisher:
Elsevier
Journal:
Tetrahedron Letters More from this journal
Volume:
74
Article number:
153151
Publication date:
2021-05-05
Acceptance date:
2021-05-01
DOI:
ISSN:
0040-4039


Language:
English
Keywords:
Pubs id:
1174043
Local pid:
pubs:1174043
Deposit date:
2021-05-04

Terms of use



Views and Downloads






If you are the owner of this record, you can report an update to it here: Report update to this record

TO TOP