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A comparison of the immunogenicity of intravenous BAT1806, a tocilizumab biosimilar, and its reference product

Abstract:

Introduction: Biosimilars need to demonstrate similarity in terms of quality, pharmacokinetics (PK), efficacy, safety and immunogenicity. Here we report the outcome of a comprehensive evaluation of the immunogenicity of the biosimilar BAT1806 compared with tocilizumab reference product (TCZ).

Methods: A post-hoc analysis of study BAT1806-001-CR, a comparative PK study in healthy male volunteers (n = 129), and BAT1806-002-CR, a phase III, 52-week trial in patients with rheumatoid arthritis (n = 621). Anti-drug antibodies (ADA), ADA titres, and neutralising ADA were measured, and their impact on PK, safety, and efficacy parameters were assessed.

Results: In BAT1806-001-CR, treatment-induced ADA were observed in 37.8% of participants for the BAT1806 group, 28.6% for the EU-sourced TCZ group and 31.0% for the US-sourced TCZ group, without impact on PK and safety. In BAT1806-002-CR after 52 weeks, 28.2% of participants in the BAT1806 group developed treatment-induced ADA, compared with 24.0% in the TCZ group and 19.7% of participants who initiated TCZ and switched to BAT1806 at week 24. ADA-positive participants reported lower geometric mean serum tocilizumab trough concentrations than ADA-negative participants in all treatment groups. ADA-positive participants achieved similar efficacy outcomes to ADA-negative participants in all treatment groups. ADA were not associated with an incremental risk of treatment-emergent adverse events or hypersensitivity in any treatment group.

Conclusions: The results of these post hoc analyses did not indicate any clinically relevant differences in the immunogenicity profile of intravenously administered BAT1806 compared with TCZ.

Trial registration: ClinicalTrials.gov identifiers, NCT03606876, NCT03830203

Publication status:
Published
Peer review status:
Peer reviewed

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Publisher copy:
10.1007/s40744-025-00760-y

Authors


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Institution:
University of Oxford
Division:
MSD
Department:
NDORMS
Sub department:
Botnar Research Centre
Oxford college:
St Peter's College
Role:
Author
ORCID:
0000-0001-7766-6167


Publisher:
Springer
Journal:
Rheumatology and Therapy More from this journal
Volume:
12
Issue:
3
Pages:
529-546
Publication date:
2025-04-08
Acceptance date:
2025-03-18
DOI:
EISSN:
2198-6584
ISSN:
2198-6576


Language:
English
Keywords:
Pubs id:
2096669
Local pid:
pubs:2096669
Deposit date:
2025-03-21

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