Journal article

A novel approach to 3-methylindoles by a Heck/cyclization/isomerization process.

Abstract:: A novel synthesis of 3-methylindoles from chlorotriflates through a Heck reaction, carbamate/aryl chloride coupling, and isomerization sequence is presented. The three-step sequence is highly efficient and general, enabling the regiocontrolled synthesis of substituted indoles in short order.

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APA Style

Baxter, C., Cleator, E., Alam, M., Davies, A., Goodyear, A., & O'Hagan, M. (2010). A novel approach to 3-methylindoles by a Heck/cyclization/isomerization process. Org Lett, 12(4), 668–671.

MLA Style

Baxter, C, et al. “A Novel Approach to 3-Methylindoles by a Heck/Cyclization/Isomerization Process.” Org Lett, vol. 12, no. 4, 2010, pp. 668–71.

Chicago Style

Baxter, C, E Cleator, M Alam, A Davies, A Goodyear, and M O'Hagan. 2010. “A Novel Approach to 3-Methylindoles by a Heck/Cyclization/Isomerization Process.” Org Lett 12 (4): 668–71.
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Publisher copy:: 10.1021/ol902636v

Authors

+ Baxter, C More by this author

Role:: Author

+ Cleator, E More by this author

Role:: Author

+ Alam, M More by this author

Role:: Author

+ Davies, A More by this author

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+ Goodyear, A More by this author

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Journal:: Org Lett More from this journal
Volume:: 12
Issue:: 4
Pages:: 668-671
Publication date:: 2010-02-19
DOI:: 10.1021/ol902636v
EISSN:: 1523-7052
ISSN:: 1523-7060

Language:: English
Keywords:: Skatole

Mesylates

Hydrocarbons, Chlorinated

Cyclization

Catalysis

Combinatorial Chemistry Techniques

Molecular Structure
UUID:: uuid:a2479168-3eb8-4212-a0b9-d0b4a4cb46d3
Local pid:: pubs:410766
Source identifiers:: 410766
Deposit date:: 2013-11-16
ARK identifier:: ark:/29072/ora_a24791683eb84212a0b9d0b4a4cb46d3

Terms of use

Copyright date:: 2010

Licence:: Terms and Conditions of Use for Oxford University Research Archive

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