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Modes of cell death induced by tetrahydroisoquinoline-based analogs in MDA-MB-231 breast and A549 lung cancer cell lines

Abstract:
Background: A and B rings of the steroidal microtubule disruptor, 2-methoxyestradiol, and its analogs can be mimicked with a tetrahydroisoquinoline (THIQ) core. THIQs are cytotoxic agents with potential anticancer activities. The aim of this in vitro study was to investigate the modes of cell death induced by four nonsteroidal THIQ-based analogs, such as STX 2895, STX 3329, STX 3451 and STX 3450, on MDA-MB-231 metastatic breast and A549 epithelial lung carcinoma cells. Expand abstract
Publication status:
Published
Peer review status:
Peer reviewed

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Publisher copy:
10.2147/DDDT.S152718

Authors


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Institution:
University of Oxford
Division:
Medical Sciences Division
Department:
Pharmacology
Role:
Author
More by this author
Institution:
University of Oxford
Division:
MSD
Department:
Pharmacology
Role:
Author
More from this funder
Funding agency for:
Potter, B
Grant:
Senior Investigator (grant 101010
Medical Research Council of South Africa More from this funder
Struwig-Germeshuysen Cancer Research Trust of South Africa More from this funder
National Research Foundation More from this funder
Cancer Association of South Africa More from this funder
Publisher:
Dove Medical Press Publisher's website
Journal:
Drug Design, Development and Therapy Journal website
Volume:
2018:12
Pages:
1881—1904
Publication date:
2018-06-25
Acceptance date:
2018-03-27
DOI:
ISSN:
1177-8881
Keywords:
Pubs id:
pubs:831923
UUID:
uuid:8db3edea-ae43-40c7-9d22-0905bfb65218
Local pid:
pubs:831923
Source identifiers:
831923
Deposit date:
2018-04-20

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