Journal article
Palladium-catalyzed desulfinative cross-couplings
- Abstract:
- The Suzuki–Miyaura reaction has undeniably revolutionized the art of synthesis, particularly in the pharmaceutical industry. However, the coupling of 2-pyridine boronic acids has long remained a challenge. In this context, our laboratory has recently reported the use of pyridyl and other heteroaryl sulfinate salts as efficient alternatives to boron reagents. This new reaction successfully yields industrially relevant building blocks, the synthesis of which would be challenging using classic boron-based nucleophiles.
- Publication status:
- Published
- Peer review status:
- Peer reviewed
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- Files:
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(Preview, Accepted manuscript, 417.9KB, Terms of use)
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- Publisher copy:
- 10.1016/j.trechm.2020.04.004
Authors
- Publisher:
- Cell Press
- Journal:
- Trends in Chemistry More from this journal
- Volume:
- 2
- Issue:
- 9
- Pages:
- 865-866
- Publication date:
- 2020-05-05
- Acceptance date:
- 2020-04-08
- DOI:
- ISSN:
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2589-7209
- Language:
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English
- Keywords:
- Pubs id:
-
1100189
- Local pid:
-
pubs:1100189
- Deposit date:
-
2020-04-15
Terms of use
- Copyright holder:
- Elsevier Inc.
- Copyright date:
- 2020
- Rights statement:
- © 2020 Elsevier Inc. All rights reserved.
- Notes:
- This is the accepted manuscript version of the article. The final version is available online from Elsevier at: https://doi.org/10.1016/j.trechm.2020.04.004
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