Journal article

Templated scaffolds of cis- and trans-tetrahydrofuran gamma-amino acids: gamma-azido-beta-hydroxy-tetrahydrofuran-2-carboxylates from pentono-delta-lactones

Abstract:: Short syntheses of enantiomeric templated scaffolds of cis- and trans-tetrahydrofuran γ-amino acids from pentono-δ-lactones derived from arabinose and ribose are reported; an unexpectedly efficient synthesis of a templated tetrahydrofuran β-amino acid by azide displacement of a triflate β to an ester function proceeds with remarkably little elimination. These materials should allow evaluation of such peptidomimetics to induce predisposition towards secondary structures. © 2003 Elsevier Ltd. All rights reserved.

Publication status:: Published

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APA Style

Sanjayan, G., Stewart, A., Hachisu, S., Gonzalez, R., Watterson, M., & Fleet, G. (2003). Templated scaffolds of cis- and trans-tetrahydrofuran gamma-amino acids: gamma-azido-beta-hydroxy-tetrahydrofuran-2-carboxylates from pentono-delta-lactones. TETRAHEDRON LETTERS, 44(31), 5847–5851.

MLA Style

Sanjayan, G, et al. “Templated Scaffolds of Cis- and Trans-Tetrahydrofuran Gamma-Amino Acids: Gamma-Azido-Beta-Hydroxy-Tetrahydrofuran-2-Carboxylates from Pentono-Delta-Lactones.” TETRAHEDRON LETTERS, vol. 44, no. 31, 2003, pp. 5847–51.

Chicago Style

Sanjayan, G, A Stewart, S Hachisu, R Gonzalez, M Watterson, and G Fleet. 2003. “Templated Scaffolds of Cis- and Trans-Tetrahydrofuran Gamma-Amino Acids: Gamma-Azido-Beta-Hydroxy-Tetrahydrofuran-2-Carboxylates from Pentono-Delta-Lactones.” TETRAHEDRON LETTERS 44 (31): 5847–51.
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Publisher copy:: 10.1016/S0040-4039(03)01415-1

Authors

+ Sanjayan, G More by this author

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+ Stewart, A More by this author

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+ Hachisu, S More by this author

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+ Gonzalez, R More by this author

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+ Watterson, M More by this author

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Journal:: TETRAHEDRON LETTERS More from this journal
Volume:: 44
Issue:: 31
Pages:: 5847-5851
Publication date:: 2003-07-28
DOI:: 10.1016/S0040-4039(03)01415-1
ISSN:: 0040-4039

Language:: English
Pubs id:: pubs:38707
UUID:: uuid:08f7ea8c-51f5-4c01-a6ee-1555974a94ba
Local pid:: pubs:38707
Source identifiers:: 38707
Deposit date:: 2012-12-19
ARK identifier:: ark:/29072/ora_08f7ea8c51f54c01a6ee1555974a94ba

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Copyright date:: 2003

Licence:: Terms and Conditions of Use for Oxford University Research Archive

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