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Journal article

The fragment molecular orbital method reveals new insight into the chemical nature of GPCR-ligand interactions

Abstract:

Our interpretation of ligand–protein interactions is often informed by high-resolution structures, which represent the cornerstone of structure-based drug design. However, visual inspection and molecular mechanics approaches cannot explain the full complexity of molecular interactions. Quantum Mechanics approaches are often too computationally expensive, but one method, Fragment Molecular Orbital (FMO), offers an excellent compromise and has the potential to reveal key interactions that would...

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Publication status:
Published
Peer review status:
Peer reviewed

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Publisher copy:
10.1021/acs.jcim.5b00644

Authors


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Institution:
University of Oxford
Division:
MSD
Department:
Biochemistry
Role:
Author
Publisher:
American Chemical Society
Journal:
Journal of Chemical Information and Modeling More from this journal
Volume:
56
Issue:
1
Pages:
159-172
Publication date:
2015-12-07
DOI:
EISSN:
1549-960X
ISSN:
1549-9596
Language:
English
Pubs id:
pubs:587370
UUID:
uuid:e46e7d6d-0eda-4f95-8ab7-393e83d6f2f7
Local pid:
pubs:587370
Source identifiers:
587370
Deposit date:
2016-03-14

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