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Enantioselective synthesis of 4- and 6-azaindolines by a cation-directed cyclization

Abstract:
Functionalized 4- and 6-azaindolines are accessible with high levels of enantioselectivity by the cation-directed cyclization of aminopyridine-derived imines via phase-transfer catalysis. The extension of this methodology to diastereoselective cyclizations is also described.
Publication status:
Published
Peer review status:
Peer reviewed

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Publisher copy:
10.1021/acs.orglett.6b02744

Authors


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Institution:
University of Oxford
Division:
MPLS
Department:
Chemistry
Sub department:
Organic Chemistry
Role:
Author
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Name:
Engineering and Physical Sciences Research Council
Grant:
EP/I003398/1
More from this funder
Name:
European Research Council
Grant:
Seventh Framework Programme (FP7/2007–2013)/ERC grant agreement no. 259056
Publisher:
American Chemical Society
Journal:
Organic Letters More from this journal
Volume:
18
Issue:
20
Pages:
5372–5375
Publication date:
2016-01-01
Acceptance date:
2016-10-03
DOI:
EISSN:
1523-7052
ISSN:
1523-7060
Pubs id:
pubs:647888
UUID:
uuid:aada17a9-37c1-4246-8623-e2ff5788a88c
Local pid:
pubs:647888
Source identifiers:
647888
Deposit date:
2016-10-04

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