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Peroxynitrite activated drug conjugate systems based on a coumarin scaffold toward the application of theranostics

Abstract:

Two novel drug-conjugates based on a “coumarin linker” have been designed for the synergic release of a therapeutic agent and fluorescent probe for the potential application of theranostics. The drug conjugates; CC-RNS and CI-RNS were designed to be activated by reactive oxygen species or reactive nitrogen species (ROS/RNS). The fluorescence OFF-ON response was triggered by the peroxynitrite-mediated transformation of a boronic acid pinacol ester to a phenol moiety with simultaneous release o...

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Publication status:
Published
Peer review status:
Peer reviewed

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Publisher copy:
10.3389/fchem.2019.00775

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Institution:
University of Oxford
Division:
MPLS Division
Department:
Chemistry
Department:
Unknown
Role:
Author
Publisher:
Frontiers Media Publisher's website
Journal:
Frontiers in Chemistry Journal website
Volume:
7
Article number:
775
Publication date:
2019-12-05
Acceptance date:
2019-10-25
DOI:
ISSN:
2296-2646
Pmid:
31867305
Language:
English
Keywords:
Pubs id:
pubs:1082182
UUID:
uuid:882611d2-c7fb-4abc-928e-ee6fbfaccff4
Local pid:
pubs:1082182
Source identifiers:
1082182
Deposit date:
2020-01-16

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