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One-pot three-component sulfone synthesis exploiting palladium-catalysed aryl halide aminosulfonylation

Abstract:

A palladium-catalysed aminosulfonylation process is used as the key-step in a one-pot, three-component sulfone synthesis. The process combines aryl-, heteroaryl- and alkenyl iodides with a sulfonyl unit and an electrophilic coupling fragment. The sulfonyl unit is delivered in the form of an aminosulfonamide, which then serves as a masked sulfinate. The sulfinate is combined, in situ, with an electrophilic coupling partner, such as a benzylic, allylic or alkyl halide, an electron-poor arene, o...

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Publication status:
Published

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Publisher copy:
10.1039/c3sc52332b

Authors


Richards-Taylor, CS More by this author
Blakemore, DC More by this author
Willis, MC More by this author
Journal:
CHEMICAL SCIENCE
Volume:
5
Issue:
1
Pages:
222-228
Publication date:
2014
DOI:
EISSN:
2041-6539
ISSN:
2041-6520
URN:
uuid:49bf6ab9-0d94-44dc-b426-c1884fa61a5c
Source identifiers:
443402
Local pid:
pubs:443402
Language:
English

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