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Journal article

Nilotinib-induced vasculopathy: Identification of vascular endothelial cells as a primary target site

Abstract:

The BCR/ABL1 inhibitor Nilotinib is increasingly used to treat patients with chronic myeloid leukemia (CML). Although otherwise well-tolerated, Nilotinib has been associated with the occurrence of progressive arterial occlusive disease (AOD). Our objective was to determine the exact frequency of AOD and examine in vitro and in vivo effects of Nilotinib and Imatinib on endothelial cells to explain AOD-development. In contrast to Imatinib, Nilotinib was found to upregulate pro-atherogenic adhes...

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Publication status:
Published
Peer review status:
Peer reviewed

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Publisher copy:
10.1038/leu.2017.245

Authors


More by this author
Institution:
University of Oxford
Division:
MSD
Department:
NDM
Sub department:
Target Discovery Institute
Role:
Author
More from this funder
Grant:
F4701-B20,F4704-B20,F5404-B20,
F5412-B2
Publisher:
Springer Nature Publisher's website
Journal:
Leukemia Journal website
Volume:
31
Issue:
11
Pages:
2388–2397
Publication date:
2017-09-08
Acceptance date:
2017-07-17
DOI:
EISSN:
1476-5551
ISSN:
0887-6924
Language:
English
Pubs id:
pubs:710904
UUID:
uuid:39785be9-6ad0-4d2c-829e-248797f10938
Local pid:
pubs:710904
Source identifiers:
710904
Deposit date:
2017-08-07

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