Subject
- Crystallography, X-Ray2
- Models, Molecular2
- Protein Structure, Tertiary2
- antagonists and inhibitors2
- chemistry2
- metabolism2
- pharmacology2
- Amino Acid Motifs1
- Dose-Response Relationship, Drug1
- Enzyme Inhibitors1
- Ketoglutaric Acids1
- Molecular Structure1
- Oxidoreductases, N-Demethylating1
- Piperazines1
- Protein Binding1
- Protein Kinase Inhibitors1
- Protein-Tyrosine Kinases1
- Pyrimidines1
- Stereoisomerism1
- Structure-Activity Relationship1